V2EX imatinib

Imatinib

定义 Definition

伊马替尼:一种酪氨酸激酶抑制剂(靶向抗癌药),常用于治疗慢性髓性白血病(CML)以及部分胃肠道间质瘤(GIST)等肿瘤,通过抑制异常激酶信号(如 BCR-ABL)来阻止癌细胞生长与增殖。(该词也常以商品名 Gleevec/Glivec 出现。)

发音 Pronunciation (IPA)

/mtnb/

例句 Examples

Imatinib is used to treat chronic myeloid leukemia.
伊马替尼用于治疗慢性髓性白血病。

After genetic testing confirmed a BCR-ABLpositive leukemia, the patient began imatinib therapy and achieved a deep molecular response over the following months.
基因检测证实该患者为 BCR-ABL 阳性的白血病后,开始接受伊马替尼治疗,并在随后数月内达到深度分子学缓解。

词源 Etymology

imatinib 属于国际非专利药名(INN)的命名体系:词尾 -nib 常见于“小分子抑制剂”类药物名称中,尤其多见于激酶抑制剂;其中的 -tinib 常用来指代酪氨酸激酶抑制剂(tyrosine kinase inhibitor)。前面的 ia- 部分主要用于区分具体分子,并非日常英语中可独立拆解的常用词根。

相关词 Related Words

文学与作品 Literary Works

  • 《The Emperor of All Maladies: A Biography of Cancer》(Siddhartha Mukherjee):作为癌症治疗史中的标志性案例之一,书中讨论了靶向治疗浪潮与相关药物(包括伊马替尼)的意义。
  • Blood(期刊):多篇关于 CML 与靶向治疗的经典综述和研究论文中频繁出现 imatinib
  • The New England Journal of Medicine(NEJM,期刊):发表过与 CML 靶向治疗相关的里程碑临床研究,文中常使用 imatinib
  • Nature Medicine(期刊):在靶向药物机制与临床转化研究中多次提及 imatinib
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