V2EX osimertinib

Osimertinib

定义 Definition

奥希替尼:一种第三代EGFR(表皮生长因子受体)酪氨酸激酶抑制剂(TKI)靶向药,常用于治疗携带特定 EGFR 突变的非小细胞肺癌(NSCLC),包括对部分耐药突变(如 T790M)也可能有效。(在不同国家/地区适应证与用法以医生与药品说明书为准。)

发音 Pronunciation

/osmrtnb/

例句 Examples

The doctor prescribed osimertinib for her EGFR-mutated lung cancer.
医生为她的 EGFR 突变型肺癌开具了奥希替尼。

In the trial, patients receiving osimertinib showed longer progression-free survival than those on earlier EGFR inhibitors.
在该临床试验中,使用奥希替尼的患者比使用早期 EGFR 抑制剂的患者显示出更长的无进展生存期。

词源 Etymology

osimertinib 是国际非专利药名(INN)风格的药物命名:结尾 -tinib 常见于酪氨酸激酶抑制剂类药名(tyrosine kinase inhibitor)的“词尾标记”,便于识别药物类别;前半部分 osimer- 多为区分不同药物的构词片段,本身通常不对应一个明确的日常词根含义。

相关词 Related Words

文献与作品 Literary Works

  • “Osimertinib in Untreated EGFR-Mutated Advanced NonSmall-Cell Lung Cancer”The New England Journal of Medicine,FLAURA 研究论文)
  • AURA3 研究相关论文(比较奥希替尼与化疗在耐药背景下的疗效,常见于肿瘤学权威期刊)
  • NCCN/ESMO 肺癌临床指南(多版指南中对 osimertinib 的推荐与用药位置有系统描述)
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